SCHEMBL31067662

SCHEMBL31067662

COc1cc2ncnc(Nc3ccc(NC(=O)Nc4ccc(F)cc4)cc3)c2cc1OC

nearest known ligand 0.82

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.82
KDR P35968 16/20 0.81
KIT P10721 1/20 0.72
HDAC3 O15379 1/20 0.68
HDAC4 P56524 1/20 0.68
HDAC1 Q13547 1/20 0.68
HDAC7 Q8WUI4 1/20 0.68
HDAC2 Q92769 1/20 0.68
HDAC10 Q969S8 1/20 0.68
HDAC11 Q96DB2 1/20 0.68
HDAC8 Q9BY41 1/20 0.68
HDAC6 Q9UBN7 1/20 0.68
HDAC9 Q9UKV0 1/20 0.68
HDAC5 Q9UQL6 1/20 0.68
AURKA O14965 1/20 0.68
AURKB Q96GD4 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31067733 0.91 KDR (0.80) EGFRKDRKIT
SCHEMBL5478005 0.91 EGFR (1.00) EGFRKDRAURKAAURKB
SCHEMBL31067640 0.90 KDR (0.84) EGFRKDRKITHDAC3HDAC4
SCHEMBL31067666 0.90 KDR (1.00) EGFRKDRKITAURKAAURKB
SCHEMBL31067650 0.90 KDR (0.83) EGFRKDRKITAURKAAURKB
Hydrochloric Acid SCHEMBL29623261 0.89 EGFR (1.00) EGFRKDRAURKAAURKB
Hydrochloric Acid SCHEMBL5471121 0.89 EGFR (1.00) EGFRKDRAURKAAURKB
SCHEMBL31067633 0.89 KDR (0.82) EGFRKDRKITHDAC3HDAC4
SCHEMBL31067708 0.89 KDR (0.82) EGFRKDRKITAURKAAURKB
SCHEMBL31067670 0.88 KDR (0.84) EGFRKDRKITAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530175-A PDGFR inhibitor and preparation method and application thereof 中国药科大学 2024-08-23 CN disclosed