SCHEMBL31067708

SCHEMBL31067708

COc1cc2ncnc(Nc3ccc(NC(=O)Nc4ccc(I)cc4)cc3)c2cc1OC

nearest known ligand 0.82

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.82
EGFR P00533 6/20 0.75
KIT P10721 1/20 0.72
AURKA O14965 1/20 0.68
AURKB Q96GD4 1/20 0.68
BRAF P15056 1/20 0.67
GAK O14976 1/20 0.67
RIPK2 O43353 1/20 0.67
STK10 O94804 1/20 0.67
RET P07949 1/20 0.67
FLT3 P36888 1/20 0.67
JAK3 P52333 1/20 0.67
AAK1 Q2M2I8 1/20 0.67
Q6ZSR9 Q6ZSR9 1/20 0.67
SLK Q9H2G2 1/20 0.67
IRAK4 Q9NWZ3 1/20 0.67
RPS6KA6 Q9UK32 1/20 0.67
ALK Q9UM73 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5473780 0.91 EGFR (0.78) KDREGFRGAKRIPK2STK10
SCHEMBL31067615 0.91 KDR (0.80) KDREGFRKITAURKAAURKB
SCHEMBL31067650 0.90 KDR (0.83) KDREGFRKITAURKAAURKB
SCHEMBL31067640 0.90 KDR (0.84) KDREGFRKITAURKAAURKB
SCHEMBL31067666 0.90 KDR (1.00) KDREGFRKITAURKAAURKB
Hydrochloric Acid SCHEMBL1507577 0.89 EGFR (0.78) KDREGFRGAKRIPK2STK10
SCHEMBL31067662 0.89 EGFR (0.82) KDREGFRKITAURKAAURKB
SCHEMBL31067633 0.89 KDR (0.82) KDREGFRKITAURKAAURKB
SCHEMBL31067741 0.87 KDR (0.79) KDREGFRKITAURKAAURKB
SCHEMBL31067608 0.86 KDR (0.85) KDREGFRKITAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118530175-A PDGFR inhibitor and preparation method and application thereof 中国药科大学 2024-08-23 CN disclosed