SCHEMBL31069716

SCHEMBL31069716

CN1CCN(Cc2cc(OC(F)(F)F)ccc2F)C(=O)c2cc(Br)cnc21

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 12/20 0.45
SLC6A2 P23975 2/20 0.40
SCN1A P35498 1/20 0.39
SCN4A P35499 1/20 0.39
KCNH2 Q12809 1/20 0.39
SCN5A Q14524 1/20 0.39
SCN9A Q15858 1/20 0.39
SCN2A Q99250 1/20 0.39
SCN3A Q9NY46 1/20 0.39
SCN8A Q9UQD0 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
GRM2 Q14416 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
ALKBH1 Q13686 1/20 0.35
CHRM5 P08912 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22470576 0.85 SCN1A (0.38) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL29714020 0.85 SCN1A (0.38) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL25380407 0.83 SCN1A (0.49) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL31069723 0.83 ALKBH1 (0.37) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL31069731 0.83 SCN1A (0.49) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL25438155 0.82 GRM2 (0.37) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL31069727 0.82 GRM2 (0.37) SCN1ASCN4AKCNH2SCN5ASCN9A
SCHEMBL25380390 0.78 TNIK (0.41) CACNA2D1SLC6A2SCN1ASCN4AKCNH2
SCHEMBL31069722 0.78 TNIK (0.41) CACNA2D1SLC6A2SCN1ASCN4AKCNH2
SCHEMBL31118862 0.75 SCN1A (0.55) SCN1ASCN4AKCNH2SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118556044-A Fused heterocyclic compound, preparation method thereof and application thereof in medicine 江苏恒瑞医药股份有限公司 2024-08-27 CN disclosed