SCHEMBL31095433

SCHEMBL31095433

COc1cncc(-n2cnc([N+](=O)[O-])c2)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
MAPT P10636 2/20 0.43
RIPK2 O43353 3/20 0.43
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
KAT2B Q92831 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25194557 1.00 HTR2A (0.44) HTR2AHTR2CHTR2BMAPTRIPK2
SCHEMBL25194715 0.86 HTR2A (0.48) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL25191480 0.83 HTR2A (0.54) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL25200431 0.82 KEAP1 (0.52) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL31095257 0.82 KEAP1 (0.52) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL20589447 0.81 HTR2A (0.44) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL25195386 0.81 HTR2A (0.44) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL31095519 0.81 HTR2A (0.44) HTR2AHTR2CHTR2BMAPTALDH1A1
SCHEMBL22237339 0.77 CYP2E1 (0.55) RIPK2CHRNB2CHRNA4MAOAMAOB
SCHEMBL25196835 0.77 ALDH1A1 (0.51) HTR2AHTR2CHTR2BMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119060060-A Imidazole-containing ALK2 kinase inhibitors 拜奥克里斯特制药公司 2024-12-03 CN disclosed
CN-110913855-B Imidazole-containing ALK2 kinase inhibitors 拜奥克里斯特制药公司 2024-09-03 CN disclosed