SCHEMBL31128

SCHEMBL31128

O=C(c1ccc(F)c(O)c1)c1ccc(-c2ccc(O)cc2)s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 20/20 1.00
HSD17B2 P37059 17/20 1.00
CLK1 P49759 1/20 0.56
DYRK1A Q13627 1/20 0.56
DYRK1B Q9Y463 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23443 0.88 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL23374 0.85 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL31434 0.83 HSD17B1 (0.79) HSD17B1HSD17B2CLK1DYRK1ADYRK1B
SCHEMBL24752 0.80 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL26606781 0.78 HSD17B1 (0.64) HSD17B1HSD17B2CLK1DYRK1ADYRK1B
SCHEMBL23686 0.77 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL22709 0.75 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL18186517 0.74 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL23409 0.73 HSD17B2 (0.61) HSD17B1HSD17B2
SCHEMBL23023 0.72 HSD17B1 (1.00) HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed