SCHEMBL31129042

SCHEMBL31129042

COc1cc(Oc2nccc(C)n2)ccc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.37
RAF1 P04049 5/20 0.36
MAP2K1 Q02750 5/20 0.36
SNCA P37840 1/20 0.35
EGFR P00533 2/20 0.34
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
UCHL1 P09936 1/20 0.32
TGFBR1 P36897 2/20 0.32
LIPE Q05469 1/20 0.32
USP2 O75604 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25594194 0.82 HTT (0.34) RAB9ARAF1MAP2K1SNCALIPE
SCHEMBL5899720 0.79 CA2 (0.47) SNCAEGFRUCHL1CYP1A2CYP3A4
SCHEMBL29424578 0.79 CA2 (0.47) SNCAEGFRUCHL1CYP1A2CYP3A4
SCHEMBL25591397 0.79 NPC1 (0.34) RAB9ARAF1MAP2K1LIPENPC1
SCHEMBL22658702 0.79 CA1 (0.43) SNCA
SCHEMBL30326281 0.78 CSF1R (0.39) SNCAEGFR
SCHEMBL25596616 0.78 MAP2K1 (0.32) RAF1MAP2K1LIPE
SCHEMBL31128931 0.75 ALOX5AP (0.39) EGFRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL17200314 0.75 DRD1 (0.41) RAB9ASNCAEGFRPDGFRBPDGFRA
SCHEMBL31128803 0.75 RAB9A (0.44) RAB9ARAF1MAP2K1EGFRPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024208315-A1 AROMATIC HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 中国医药研究开发中心有限公司 2024-10-10 WO disclosed