SCHEMBL3114375

SCHEMBL3114375

NCc1nc(-c2ccc(Cl)cc2)c(-c2ccc(Cl)cc2Cl)cc1CNC(=O)NCc1ccccc1F

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.58
DPP4 P27487 2/20 0.39
IDH1 O75874 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
PKM P14618 1/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EIF4E P06730 1/20 0.37
PPIA P62937 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3103553 0.92 CNR1 (0.58) CNR1IDH1MEN1KMT2ALMNA
SCHEMBL3113229 0.88 CNR1 (0.55) CNR1IDH1KMT2APKMRAB9A
SCHEMBL3110050 0.88 CNR1 (0.60) CNR1IDH1KMT2AEIF4EPPIA
SCHEMBL3104836 0.85 CNR1 (0.56) CNR1IDH1KMT2AMAPT
SCHEMBL3224422 0.85 CNR1 (0.52) CNR1IDH1KMT2A
SCHEMBL3110196 0.79 DPP4 (0.48) CNR1DPP4LMNAMAPT
SCHEMBL3713619 0.76 CNR1 (0.53) CNR1KMT2AMAPT
SCHEMBL3100296 0.74 DDR1 (0.45) CNR1DPP4LMNA
SCHEMBL13307940 0.73 CNR1 (1.00) CNR1
SCHEMBL3115945 0.72 KCNK2 (0.39) CNR1DPP4MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8362045-B2 5,6-diaryl pyridines substituted in the 2- and 3-position, preparation thereof and therapeutic use thereof SANOFI (FR) 2013-01-29 US disclosed
US-20100256202-A1 5,6-DIARYL PYRIDINES SUBSTITUTED IN THE 2- AND 3-POSITION, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2010-10-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100256202-A1 5,6-DIARYL PYRIDINES SUBSTITUTED IN THE 2- AND 3-POSITION, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF ALK, ROS1, CYP11B2 CNR1 11/4885DPP4 1949/4885IDH1 219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.