SCHEMBL3116231

SCHEMBL3116231

O=C(CCC1CCN(CCc2ccccc2)CC1)Nc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.56
CA1 P00915 1/20 0.55
CA2 P00918 1/20 0.55
CA9 Q16790 1/20 0.55
MAPT P10636 1/20 0.55
HTT P42858 1/20 0.55
CCR3 P51677 1/20 0.55
ALDH1A1 P00352 1/20 0.54
POLB P06746 1/20 0.54
LMNA P02545 1/20 0.54
KMT2A Q03164 1/20 0.54
RAB9A P51151 1/20 0.54
HTR1A P08908 1/20 0.53
DRD2 P14416 1/20 0.53
HTR2A P28223 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16653309 0.90 MAPT (0.50) SIGMAR1MAPTCCR3ALDH1A1POLB
SCHEMBL12059418 0.87 BCHE (0.66) POLBKMT2ADRD2
SCHEMBL5276400 0.87 EPHX2 (0.59) SIGMAR1CCR3HTR1ADRD2HTR2A
SCHEMBL27808768 0.82 MAPT (0.49) CA1CA2CA9MAPTHTT
SCHEMBL8016039 0.82 CCR3 (0.60) SIGMAR1CCR3HTR2A
SCHEMBL7801292 0.80 ACHE (0.59) SIGMAR1LMNA
SCHEMBL5870720 0.78 LTA4H (0.52) MAPTHTTALDH1A1POLBLMNA
SCHEMBL29086653 0.78 KLK7 (0.72) MAPTHTTALDH1A1KMT2ARAB9A
SCHEMBL29381887 0.78 CCR3 (0.75) CCR3
SCHEMBL5276763 0.78 DCUN1D1 (0.60) MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010033540-A1 CRYSTALLINE FORMS OF FENTANYL ALKALOID MALLINCKRODT INC. (US) 2010-03-25 WO claimed