SCHEMBL31190896

SCHEMBL31190896

O=Cc1cccc(-c2cn[nH]c2)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.41
AKT1 P31749 1/20 0.41
AKT2 P31751 1/20 0.41
ERN1 O75460 1/20 0.40
ROCK2 O75116 7/20 0.38
ROCK1 Q13464 6/20 0.38
DRD1 P21728 2/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
FEN1 P39748 1/20 0.35
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
INCENP Q9NQS7 1/20 0.34
TPX2 Q9ULW0 1/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
P2RX7 Q99572 1/20 0.33
ADRA1B P35368 1/20 0.33
XDH P47989 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1956753 0.83 AKT2 (0.50) PDK2AKT1AKT2ERN1ROCK2
SCHEMBL31663053 0.76 ROCK2 (0.39) PDK2AKT1AKT2ERN1ROCK2
SCHEMBL24802714 0.75 TDP1 (0.44) AKT2ERN1ROCK2ROCK1XDH
SCHEMBL4033813 0.74 KMT2A (0.46) ERN1XDH
SCHEMBL29628511 0.74 TSHR (0.46) PDK2AKT1AKT2ROCK2ROCK1
SCHEMBL29746276 0.73 ERN1 (0.34) ERN1P2RX7XDH
SCHEMBL24217030 0.72 XDH (0.36) ERN1XDH
SCHEMBL31190907 0.71 POLB (0.55) AKT1AKT2ROCK2ROCK1ADRA1D
SCHEMBL29749647 0.71 ERN1 (0.34) ERN1XDH
SCHEMBL5380089 0.71 AKT1 (0.55) PDK2AKT1AKT2ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3997096-B1 NEW HETEROCYCLIC COMPOUNDS HOFFMANN LA ROCHE (CH) 2024-08-28 EP claimed