SCHEMBL31284271

SCHEMBL31284271

COC(=O)c1ccc(C2=CCN(C(=O)OC(C)(C)C)C2)c(OC)n1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.42
PDK4 Q16654 1/20 0.41
PDE10A Q9Y233 1/20 0.38
NAMPT P43490 1/20 0.38
GRM1 Q13255 8/20 0.38
GRM5 P41594 7/20 0.38
JAK1 P23458 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HTR6 P50406 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31284146 1.00 NR1H2 (0.42) NR1H2PDK4PDE10ANAMPTGRM1
SCHEMBL20934809 0.84 PDK4 (0.42) NR1H2PDK4PDE10ANAMPTGRM1
SCHEMBL3466461 0.80 PDK4 (0.44) NR1H2PDK4PDE10ANAMPTGRM1
SCHEMBL31589595 0.79 GRM1 (0.43) NR1H2PDK4NAMPTGRM1GRM5
SCHEMBL31155284 0.79 PDE10A (0.49) PDK4PDE10ANAMPTGRM1GRM5
SCHEMBL25345866 0.79 PDE10A (0.49) PDK4PDE10ANAMPTGRM1GRM5
SCHEMBL31589298 0.79 GRM1 (0.43) NR1H2PDK4NAMPTGRM1GRM5
SCHEMBL29220909 0.78 GPR119 (0.54) NR1H2PDK4NAMPTGRM1GRM5
SCHEMBL27202971 0.77 PDK4 (0.52) PDK4PDE10ANAMPTGRM1GRM5
SCHEMBL31097527 0.77 PDK4 (0.51) PDK4NAMPTGRM1GRM5JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119176772-A Compound with Mrgpr X receptor inhibition effect and application thereof 博济医药科技股份有限公司 2024-12-24 CN disclosed