SCHEMBL3128556

SCHEMBL3128556

CS(=O)(=O)c1ccc(CC(N)=O)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.43
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRE P78334 1/20 0.41
GABRA6 Q16445 1/20 0.41
GABRG1 Q8N1C3 1/20 0.41
GABRG3 Q99928 1/20 0.41
GABRQ Q9UN88 1/20 0.41
PIK3CD O00329 1/20 0.39
PIP5K1C O60331 1/20 0.39
PIK3CB P42338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18503863 0.85 GABRP (0.54) CA2GABRPGABRDGABRA1GABRB1
SCHEMBL3121506 0.84 ALDH1A1 (0.46) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL3129950 0.83 ALDH1A1 (0.41) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL1145511 0.79 PIK3CD (0.42) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL5758401 0.79 PIK3CD (0.42) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL20489229 0.79 PIK3CD (0.39) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL29995663 0.79 PIK3CD (0.39) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL13180189 0.77 KDM4E (0.41) CA2PIK3CDPIP5K1CPIK3CBPI4KA
SCHEMBL3126015 0.75 GABRP (0.42) CA2GABRPGABRDGABRA1GABRB1
SCHEMBL2643755 0.75 PIK3CD (0.39) CA2PIK3CDPIP5K1CPIK3CBPI4KA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed