SCHEMBL3128668

SCHEMBL3128668

O=CCc1cc(Nc2nc(-c3cccnc3)c(F)s2)ccc1Oc1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 8/20 0.41
KMT2A Q03164 8/20 0.41
MAPT P10636 3/20 0.41
RAB9A P51151 4/20 0.37
ALDH1A1 P00352 2/20 0.37
PDE10A Q9Y233 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 2/20 0.35
EGFR P00533 1/20 0.35
DHODH Q02127 1/20 0.35
PTGDR2 Q9Y5Y4 4/20 0.34
GRM4 Q14833 1/20 0.34
MET P08581 1/20 0.34
CYP1A1 P04798 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP1B1 Q16678 1/20 0.34
SCN5A Q14524 1/20 0.34
SCN9A Q15858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3131583 0.92 MEN1 (0.39) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3119888 0.90 MEN1 (0.38) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL27810967 0.84 MEN1 (0.40) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3130261 0.84 MEN1 (0.62) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3117167 0.83 CHRNA7 (0.42) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3128663 0.82 MEN1 (0.43) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3127436 0.81 SGMS2 (0.37) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL27810966 0.80 MEN1 (0.40) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL28784609 0.77 MEN1 (0.42) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL3128687 0.76 MEN1 (0.56) MEN1KMT2AMAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2164846-A2 HETEROARYL SUBSTITUTED THIAZOLES AND THEIR USE AS ANTIVIRAL AGENTS. Achillion Pharmaceuticals, Inc. (US) 2010-03-24 EP claimed
WO-2008147557-A2 HETEROARYL SUBSTITUTED THIAZOLES AND THEIR USE AS ANTIVIRAL AGENTS ACHILLION PHARMACEUTICALS, INC. (US) 2008-12-04 WO claimed