SCHEMBL3132012

SCHEMBL3132012

COc1cccc(CNC(=O)Nc2ccc(-c3ccnc(N)c3)cc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 1.00
ROCK1 Q13464 8/20 0.62
CYP3A4 P08684 4/20 0.57
PRKACA P17612 3/20 0.57
NAMPT P43490 2/20 0.56
HIF1A Q16665 1/20 0.55
CYP2D6 P10635 2/20 0.55
CYP2C9 P11712 1/20 0.55
GSK3A P49840 1/20 0.55
GSK3B P49841 1/20 0.55
PRKX P51817 1/20 0.55
PRKCQ Q04759 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
AURKA O14965 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3127521 0.87 ROCK2 (1.00) ROCK2ROCK1CYP3A4PRKACANAMPT
SCHEMBL3127087 0.85 ROCK2 (0.73) ROCK2ROCK1NAMPT
SCHEMBL3120901 0.84 ROCK2 (1.00) ROCK2ROCK1NAMPTHIF1A
SCHEMBL21768820 0.82 ROCK2 (0.69) ROCK2ROCK1CYP3A4PRKACACYP2D6
SCHEMBL3249431 0.79 ROCK2 (1.00) ROCK2ROCK1NAMPTCYP2C9
SCHEMBL21768656 0.79 ROCK2 (0.65) ROCK2ROCK1CYP3A4PRKACACYP2D6
SCHEMBL1492960 0.79 CNR1 (0.66) ROCK2ROCK1CYP3A4
SCHEMBL3246062 0.78 ROCK2 (0.70) ROCK2ROCK1CYP3A4PRKACANAMPT
SCHEMBL29804102 0.77 ROCK2 (0.64) ROCK2ROCK1CYP3A4PRKACANAMPT
SCHEMBL28571017 0.77 ROCK2 (0.64) ROCK2ROCK1CYP3A4PRKACANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO disclosed