SCHEMBL29804102

SCHEMBL29804102

COc1cccc(CNC(=O)Nc2cccc(-c3ccc(C(N)=O)cc3)c2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 6/20 0.64
SMN1; SMN2 Q16637 1/20 0.57
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
PRKACA P17612 1/20 0.54
GSK3A P49840 1/20 0.54
GSK3B P49841 1/20 0.54
PRKX P51817 1/20 0.54
PRKCQ Q04759 1/20 0.54
ROCK1 Q13464 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
NAMPT P43490 2/20 0.54
PLG P00747 1/20 0.53
PLAU P00749 1/20 0.53
PLAT P00750 1/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28571017 1.00 ROCK2 (0.64) ROCK2SMN1; SMN2CYP3A4CYP2D6CYP2C9
SCHEMBL29804057 0.84 ROCK2 (0.62) ROCK2SMN1; SMN2PLAUMEN1KMT2A
SCHEMBL29804411 0.84 ROCK2 (0.56) ROCK2SMN1; SMN2GSK3BCLK4NAMPT
SCHEMBL28584102 0.84 ROCK2 (0.56) ROCK2SMN1; SMN2GSK3BCLK4NAMPT
SCHEMBL29804195 0.78 LMNA (0.66) ROCK2SMN1; SMN2ROCK1NAMPTMEN1
SCHEMBL28577264 0.78 LMNA (0.66) ROCK2SMN1; SMN2ROCK1NAMPTMEN1
SCHEMBL29804062 0.78 ROCK2 (0.63) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL28574045 0.78 ROCK2 (0.63) ROCK2CYP3A4CYP2D6CYP2C9ROCK1
SCHEMBL3127521 0.78 ROCK2 (1.00) ROCK2SMN1; SMN2CYP3A4CYP2D6CYP2C9
SCHEMBL8176742 0.78 SMN1; SMN2 (0.81) ROCK2SMN1; SMN2NAMPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112961081-B Bibenzamide urea compound and preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2022-09-13 CN claimed
CN-112961081-B Bibenzamide urea compound and preparation method and application thereof 山东第一医科大学(山东省医学科学院) 2022-09-13 CN disclosed