SCHEMBL31320126

SCHEMBL31320126

O=C(Nc1nccs1)Nc1nccc(CBr)c1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.49
PIM1 P11309 1/20 0.49
CDK2 P24941 1/20 0.49
GSK3B P49841 1/20 0.49
SMN1; SMN2 Q16637 4/20 0.47
MAPT P10636 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
CASP3 P42574 1/20 0.47
HTT P42858 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
LMNA P02545 2/20 0.44
TP53 P04637 2/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31320130 0.89 AURKA (0.50) AURKAPIM1CDK2GSK3BSMN1; SMN2
SCHEMBL31320129 0.77 SMN1; SMN2 (0.52) AURKAPIM1CDK2GSK3BSMN1; SMN2
SCHEMBL31320131 0.76 ABL1 (0.44)
SCHEMBL31320122 0.74 TYK2 (0.43) SMN1; SMN2MEN1KMT2AHTTTSHR
SCHEMBL27791809 0.67 ACP1 (0.63) SMN1; SMN2MAPTMEN1KMT2ATP53
SCHEMBL479906 0.67 ACP1 (0.63) SMN1; SMN2MEN1KMT2AHTTTP53
SCHEMBL4600722 0.66 AURKA (1.00) AURKAPIM1CDK2GSK3BSMN1; SMN2
SCHEMBL7058895 0.66 AURKA (0.61) AURKAPIM1CDK2GSK3BSMN1; SMN2
SCHEMBL17186325 0.66 KDM4E (0.60) SMN1; SMN2MAPTMEN1KMT2ATP53
SCHEMBL3524273 0.65 ACP1 (0.62) AURKAPIM1CDK2GSK3BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024240108-A1 ARYL UREA PARP1 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海海和药物研究开发股份有限公司 2024-11-28 WO disclosed