SCHEMBL31320131

SCHEMBL31320131

CCNC(=O)Nc1nccc(CBr)c1F

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.44
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
TYK2 P29597 1/20 0.37
IDO1 P14902 1/20 0.36
PIK3CA P42336 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
KIT P10721 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
MAPK1 P28482 1/20 0.35
FGFR1 P11362 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31320125 0.87 ABL1 (0.44) ABL1JAK2JAK1TYK2PIK3CA
SCHEMBL31320122 0.78 TYK2 (0.43) TYK2IDO1
SCHEMBL31320136 0.77 GAA (0.51) ABL1
SCHEMBL31320126 0.76 AURKA (0.49)
SCHEMBL31320119 0.73 MAPK1 (0.37) ABL1MAPK1
SCHEMBL31320118 0.70 ABL1 (0.41) ABL1JAK2JAK1TYK2PIK3CA
SCHEMBL31320133 0.69 GRM4 (0.34) ABL1MAPK1
SCHEMBL23694234 0.69 MEN1 (0.38) MAPK1
SCHEMBL31032965 0.69 KDR (0.41) ABL1PIK3CAMAPK8MAPK9MAPK10
SCHEMBL12410296 0.69 ABL1 (0.54) ABL1MKNK2FGFR1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024240108-A1 ARYL UREA PARP1 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海海和药物研究开发股份有限公司 2024-11-28 WO disclosed