SCHEMBL31320122

SCHEMBL31320122

O=C(Nc1nccc(CBr)c1F)NC1CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.43
DRD2 P14416 1/20 0.42
DRD4 P21917 1/20 0.42
DRD3 P35462 1/20 0.42
EPHX2 P34913 3/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 1/20 0.39
NPC1 O15118 5/20 0.39
RAB9A P51151 4/20 0.39
EPHX1 P07099 2/20 0.39
TSHR P16473 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
IDO1 P14902 1/20 0.37
HTT P42858 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31320131 0.78 ABL1 (0.44) TYK2IDO1
SCHEMBL31320126 0.74 AURKA (0.49) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL24857980 0.69 GSK3B (0.47) TYK2KMT2AMEN1
SCHEMBL31320125 0.66 ABL1 (0.44) TYK2
SCHEMBL31100376 0.65 CRBN (0.49)
SCHEMBL17607004 0.65 HTT (0.54) DRD2DRD4DRD3KMT2AMEN1
SCHEMBL31032862 0.65 DRD2 (0.50) DRD2DRD4DRD3KMT2AMEN1
SCHEMBL23694234 0.64 MEN1 (0.38) KMT2AMEN1ALDH1A1TSHR
SCHEMBL31320119 0.63 MAPK1 (0.37) NPC1RAB9ASMN1; SMN2
SCHEMBL26613698 0.63 L3MBTL1 (0.42) ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024240108-A1 ARYL UREA PARP1 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF 上海海和药物研究开发股份有限公司 2024-11-28 WO disclosed