SCHEMBL31325366

SCHEMBL31325366

COC=Cc1ccc(Br)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP1B1 Q16678 1/20 0.40
GPR183 P32249 1/20 0.36
NFE2L2 Q16236 5/20 0.35
APLNR P35414 2/20 0.35
DGAT1 O75907 1/20 0.34
EGFR P00533 1/20 0.34
RET P07949 1/20 0.34
KIF5B P33176 1/20 0.34
KDR P35968 1/20 0.34
ACHE P22303 1/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
KDM1A O60341 2/20 0.33
KDM1B Q8NB78 1/20 0.33
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1428556 1.00 CYP1A1 (0.40) CYP1A1CYP1A2CYP1B1GPR183NFE2L2
SCHEMBL1428554 1.00 CYP1A1 (0.40) CYP1A1CYP1A2CYP1B1GPR183NFE2L2
SCHEMBL1276360 0.85 NFE2L2 (0.39) GPR183NFE2L2ALDH1A1MAPTAMY1A
SCHEMBL2142490 0.85 NFE2L2 (0.39) GPR183NFE2L2ALDH1A1MAPTAMY1A
SCHEMBL21352123 0.81 APLNR (0.36) CYP1A1CYP1A2CYP1B1GPR183APLNR
SCHEMBL12732543 0.79 GPR183 (0.39) CYP1A1CYP1A2CYP1B1GPR183NFE2L2
SCHEMBL31573785 0.78 APP (0.37)
SCHEMBL31573606 0.78 APP (0.37)
SCHEMBL31573688 0.78 APP (0.37)
SCHEMBL23888923 0.77 CYP1A1 (0.37) CYP1A1CYP1A2CYP1B1GPR183NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4737437-A1 DPP1 INHIBITOR INTERMEDIATE, AND PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINES Haisco Pharmaceuticals Pte. Ltd. (SG) 2026-05-06 EP disclosed
WO-2025002093-A1 DPP1 INHIBITOR INTERMEDIATE, AND PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINES 西藏海思科制药有限公司 2025-01-02 WO disclosed