SCHEMBL31353069

SCHEMBL31353069

O=c1[nH]c2cc(Br)ccc2n2cncc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.60
PDE5A O76074 2/20 0.46
PDE9A O76083 2/20 0.46
GABRA5 P31644 2/20 0.43
GABRA1 P14867 1/20 0.43
METAP2 P50579 1/20 0.37
LCK P06239 1/20 0.36
PARP1 P09874 3/20 0.35
AURKA O14965 2/20 0.34
POLB P06746 1/20 0.34
CHEK1 O14757 2/20 0.34
GSK3B P49841 2/20 0.34
CHEK2 O96017 1/20 0.34
CDK1 P06493 1/20 0.34
PRKDC P78527 1/20 0.34
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29235466 0.88 TP53 (0.46) TP53PDE5APDE9AGABRA5GABRA1
SCHEMBL31377494 0.78 GABRA5 (0.42) TP53GABRA5PARP1POLBCHEK1
SCHEMBL4763948 0.78 PARP1 (0.59) GABRA5GABRA1PARP1POLBCHEK1
SCHEMBL30095396 0.78 PARP1 (0.59) GABRA5GABRA1PARP1POLBCHEK1
SCHEMBL31353079 0.77 GRIN2D (0.36) TP53GABRA5GABRA1LCK
SCHEMBL31026839 0.77 TP53 (0.35) TP53PDE5APDE9AGABRA5GABRA1
SCHEMBL29235228 0.77 GRIA1 (0.46) TP53PDE5APDE9A
SCHEMBL29235288 0.77 GRIN2D (0.37) TP53GABRA5GABRA1LCK
SCHEMBL7983698 0.77 TP53 (0.35) TP53PDE5APDE9AGABRA5GABRA1
SCHEMBL4036186 0.76 PARP1 (0.42) GABRA5GABRA1PARP1POLBCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119143752-A Aminoquinoline derivative, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2024-12-17 CN disclosed