SCHEMBL3135680

SCHEMBL3135680

O=C1c2ccccc2C(=O)N1C/C=C1\CCN(OC(=O)C(F)(F)F)CC1F

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.32
GAA P10253 2/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32
ACHE P22303 1/20 0.32
CASP3 P42574 1/20 0.32
CA12 O43570 1/20 0.32
CA9 Q16790 1/20 0.32
MAPK1 P28482 2/20 0.31
KMT2A Q03164 3/20 0.31
MEN1 O00255 2/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3132048 0.82 CA12 (0.35) HSD17B10GAALMNAPKMCASP3
SCHEMBL3559325 0.79 MAPK1 (0.40) HSD17B10GAALMNACA12CA9
SCHEMBL13315704 0.78 PDK4 (0.41) PKM
SCHEMBL3126790 0.77 ALDH1A1 (0.35) HSD17B10GAALMNAPKMACHE
SCHEMBL3135732 0.77 ALDH1A1 (0.35) HSD17B10GAALMNAPKMACHE
Trifluoroacetic Acid SCHEMBL3135672 0.72 KEAP1 (0.36) CASP3CA12CA9KMT2AMEN1
Trifluoroacetic Acid SCHEMBL3135667 0.72 KEAP1 (0.36) CASP3CA12CA9KMT2AMEN1
SCHEMBL3138673 0.70 ALDH1A1 (0.44) HSD17B10GAALMNAACHEMAPK1
SCHEMBL13349422 0.69 PDK4 (0.41) HSD17B10PKM
SCHEMBL3556756 0.69 MAPK1 (0.40) HSD17B10GAALMNACA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056633-A2 7-AMINO ALKYLIDENYL-HETEROCYCLIC QUINOLONES AND NAPHTHYRIDONES JANSSEN PHARMACEUTICA NV (BE) 2010-05-20 WO disclosed