SCHEMBL3136134

SCHEMBL3136134

O=C(NCc1ccccc1Cl)OC1CC(c2cc(NC(=O)C3CCCO3)[nH]n2)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.56
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
GAA P10253 1/20 0.38
JAK2 O60674 1/20 0.38
TYK2 P29597 1/20 0.38
HPGD P15428 5/20 0.38
ALDH1A1 P00352 4/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3122474 1.00 PKM (0.56) PKMNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3122481 1.00 PKM (0.56) PKMNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3121250 0.91 PKM (0.43) PKMNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3133412 0.91 PKM (0.43) PKMNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3121238 0.91 PKM (0.43) PKMNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3122362 0.90 HPGD (0.49) PKMNPC1RAB9ASMN1; SMN2ADORA3
SCHEMBL3122401 0.90 HPGD (0.49) PKMNPC1RAB9ASMN1; SMN2ADORA3
SCHEMBL3122380 0.90 HPGD (0.49) PKMNPC1RAB9ASMN1; SMN2ADORA3
SCHEMBL3131648 0.89 ADORA3 (0.45) PKMNPC1RAB9ASMN1; SMN2LMNA
SCHEMBL3133082 0.89 ADORA3 (0.45) PKMNPC1RAB9ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689721-B1 AMINOPYRAZOLE DERIVATIVES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2010-07-14 EP claimed
US-7671072-B2 Aminopyrazole derivatives as GSK-3 inhibitors PFIZER INC. (US) 2010-03-02 US claimed