Benzoxazolinone

Benzoxazolinone

SCHEMBL3136432

NC(=O)C1CNC(=O)O1.O=c1[nH]c2ccccc2o1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGT O15294 1/20 0.55
SMYD3 Q9H7B4 1/20 0.36
F2 P00734 1/20 0.36
CFD P00746 1/20 0.36
IL4I1 Q96RQ9 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
CREBBP Q92793 1/20 0.35
GAA P10253 1/20 0.34
PSMB8 P28062 1/20 0.34
NOS1 P29475 4/20 0.34
NOS3 P29474 3/20 0.34
NOS2 P35228 3/20 0.34
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
ADRA2A P08913 1/20 0.34
TSHR P16473 1/20 0.34
THPO P40225 1/20 0.34
BLM P54132 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzoxazolinone SCHEMBL17260632 0.80 OGT (0.81) OGTSMYD3F2CFDIL4I1
Benzoxazolinone SCHEMBL27217390 0.77 OGT (0.75) OGTSMYD3F2CFDIL4I1
Benzoxazolinone SCHEMBL3927631 0.74 OGT (1.00) OGTF2CFDIL4I1ALDH1A1
Benzoxazolinone SCHEMBL9110846 0.74 OGT (1.00) OGTF2CFDIL4I1ALDH1A1
Benzoxazolinone SCHEMBL29475399 0.74 OGT (1.00) OGTF2CFDIL4I1ALDH1A1
Benzoxazolinone SCHEMBL19555 0.74 OGT (1.00) OGTF2CFDIL4I1ALDH1A1
Benzoxazolinone SCHEMBL3650873 0.73 OGT (0.95) OGTF2CFDIL4I1ALDH1A1
Benzoxazolinone SCHEMBL28920994 0.73 OGT (0.95) OGTF2CFDIL4I1ALDH1A1
Benzoxazolinone SCHEMBL28598217 0.73 OGT (0.95) OGTF2CFDIL4I1ALDH1A1
SCHEMBL3144405 0.70 USP2 (0.31) ALDH1A1USP2HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645781-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER INC (US) 2010-01-12 US disclosed
US-20070015801-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives THOMAS RICHARD C 2007-01-18 US disclosed
US-7141588-B2 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PFIZER, INC. (US) 2006-11-28 US disclosed
EP-1478629-B1 N-ARYL-2-OXAZOLIDINONE-5-CARBOXAMIDES AND THEIR DERIVATIVES AND THEIR USE AS ANTIBACTERIALS PHARMACIA & UPJOHN CO LLC (US) 2006-10-11 EP disclosed
US-6919329-B2 N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives PHARMACIA & UPJOHN COMPANY (US) 2005-07-19 US disclosed
EP-1478629-A1 N-ARYL-2-OXAZOLIDINONE-5-CARBOXAMIDES AND THEIR DERIVATIVES AND THEIR USE AS ANTIBACTERIALS PHARMACIA & UPJOHN COMPANY (US) 2004-11-24 EP disclosed
US-20040147760-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives PHARMACIA & UPJOHN COMPANY 2004-07-29 US disclosed
US-20040044052-A1 N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives PHARMACIA & UPJOHN COMPANY 2004-03-04 US disclosed
WO-2003072553-A1 N-ARYL-2-OXAZOLIDINONE-5-CARBOXAMIDES AND THEIR DERIVATES AND THEIR USE AS ANTIBACTERIALS PHARMACIA & UPJOHN COMPANY (US) 2003-09-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040147760-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives OXA1L, AADAC, MT-ND5 OGT 239/4885SMYD3 3370/4885F2 4753/4885
US-20040044052-A1 N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives OXA1L, AADAC, MT-ND5 OGT 239/4885SMYD3 3370/4885F2 4753/4885
US-20070015801-A1 N-aryl-2-oxazolidinone-5-carboxamides and their derivatives OXA1L, AADAC, MT-ND5 OGT 239/4885SMYD3 3370/4885F2 4753/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.