SCHEMBL3137352

SCHEMBL3137352

COC(=O)c1cc(OC(C)=O)c2ccccc2c1-c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 3/20 0.49
TSHR P16473 2/20 0.44
HTT P42858 2/20 0.44
CFD P00746 1/20 0.43
KDM4E B2RXH2 5/20 0.43
HPGD P15428 4/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 2/20 0.40
ALDH1A1 P00352 4/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
HSD17B10 Q99714 3/20 0.39
ESR1 P03372 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
HMGB1 P09429 1/20 0.39
GGT1 P19440 1/20 0.39
PTGS1 P23219 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9899201 0.90 NR4A2 (0.46) SLC6A3TSHRHTTCFDKDM4E
SCHEMBL1009498 0.90 TSHR (0.48) SLC6A3TSHRHTTCFDKDM4E
SCHEMBL3151462 0.88 MAPK8 (0.47) SLC6A3CFDKMT2AALDH1A1NR4A2
SCHEMBL27165405 0.87 CFD (0.41) SLC6A3HTTCFDKDM4EHPGD
SCHEMBL174812 0.86 CFD (0.43) SLC6A3TSHRCFDKDM4EHPGD
SCHEMBL8511704 0.86 BACE1 (0.44) SLC6A3HTTCFDKDM4EKMT2A
SCHEMBL25876669 0.86 BACE1 (0.44) SLC6A3HTTCFDKDM4EHPGD
SCHEMBL1334088 0.84 DHODH (0.53) TSHRHTTKDM4EHPGDKMT2A
SCHEMBL27165414 0.84 CFD (0.39) SLC6A3CFDKDM4EHPGDTP53
SCHEMBL9899016 0.82 NR4A2 (0.50) SLC6A3TSHRCFDKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963896-B1 PHOTOCHROMIC MATERIALS HAVING ELECTRON-WITHDRAWING SUBSTITUENTS TRANSITIONS OPTICAL INC (US) 2010-02-10 EP disclosed
US-7556751-B2 Photochromic materials having electron-withdrawing substituents TRANSITIONS OPTICAL, INC. (US) 2009-07-07 US disclosed
EP-1963896-A1 PHOTOCHROMIC MATERIALS HAVING ELECTRON-WITHDRAWING SUBSTITUENTS TRANSITIONS OPTICAL, INC. (US) 2008-09-03 EP disclosed
WO-2007073462-A1 PHOTOCHROMIC MATERIALS HAVING ELECTRON-WITHDRAWING SUBSTITUENTS TRANSITIONS OPTICAL, INC. (US) 2007-06-28 WO disclosed
US-20070138449-A1 Photochromic materials having electron-withdrawing substituents TRANSITIONS OPTICAL LIMITED (IE) 2007-06-21 US disclosed