SCHEMBL31410

SCHEMBL31410

COc1ccc(C(=O)c2nc3ccc(OC)cc3s2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.73
HSD17B2 P37059 2/20 0.73
SCD O00767 7/20 0.62
NPC1 O15118 4/20 0.62
RAB9A P51151 4/20 0.62
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
MAPT P10636 3/20 0.58
PDK1 Q15118 1/20 0.56
MAOA P21397 1/20 0.56
MAOB P27338 1/20 0.56
CYP1A2 P05177 3/20 0.56
CYP3A4 P08684 3/20 0.56
CYP2C19 P33261 3/20 0.56
HTT P42858 1/20 0.56
DYRK1A Q13627 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404873 0.93 HSD17B1 (0.72) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL8402858 0.93 HSD17B1 (0.69) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL8405382 0.92 HSD17B1 (0.67) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL8403873 0.92 HSD17B1 (0.67) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL31119 0.91 HSD17B1 (0.65) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL8402835 0.88 SCD (0.68) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL30921 0.86 HSD17B1 (0.73) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL23147 0.86 HSD17B1 (0.67) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL11007700 0.86 KMT2A (0.66) HSD17B1HSD17B2SCDNPC1RAB9A
SCHEMBL30222 0.85 HSD17B1 (0.79) HSD17B1HSD17B2SCDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
US-5900426-A ANTILIPEMIC AGENTS NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1999-05-04 US disclosed
EP-0735029-B1 Benzothiazole derivatives NIPPON ZOKI PHARMACEUTICAL CO (JP) 1998-06-03 EP disclosed
EP-0735029-A1 Benzothiazole derivatives NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1996-10-02 EP disclosed