SCHEMBL31427140

SCHEMBL31427140

COc1cccc(CN2Cc3ccc(Br)cc3N(C)C[C@@H]2C)c1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.43
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
MDM2 Q00987 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
CMA1 P23946 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
LPO P22079 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25197107 1.00 HRH3 (0.43) HRH3LMNAHTTMDM2SIGMAR1
SCHEMBL31427148 1.00 HRH3 (0.43) HRH3LMNAHTTMDM2SIGMAR1
SCHEMBL25215671 1.00 HRH3 (0.43) HRH3LMNAHTTMDM2SIGMAR1
SCHEMBL25215892 0.83 ROCK2 (0.47) HRH3SIGMAR1KDM4EALDH1A1
SCHEMBL31427147 0.83 ROCK2 (0.47) HRH3SIGMAR1KDM4EALDH1A1
SCHEMBL31427146 0.83 ROCK2 (0.47) HRH3SIGMAR1KDM4EALDH1A1
SCHEMBL25211576 0.83 ROCK2 (0.47) HRH3SIGMAR1KDM4EALDH1A1
SCHEMBL31427144 0.80 ROCK2 (0.51) HRH3SIGMAR1KDM4EALDH1A1
SCHEMBL25198645 0.74 RIPK1 (0.39)
SCHEMBL25198448 0.74 BRD4 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178337-B Benzodiazepine compounds and their use as Rho kinase inhibitors 成都奥睿药业有限公司 2025-04-25 CN disclosed