SCHEMBL3143028

SCHEMBL3143028

Cc1ncc(OCC2(CN)CC2)cc1-c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA7 P36544 1/20 0.39
BACE1 P56817 2/20 0.35
APP P05067 1/20 0.35
MAP4K4 O95819 4/20 0.34
KMT2A Q03164 7/20 0.34
MEN1 O00255 6/20 0.34
NPC1 O15118 2/20 0.33
HPGD P15428 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3773920 0.99 CHRNB4 (0.39) CHRNB4CHRNA3CHRNA7BACE1APP
SCHEMBL3147035 0.89 ABL1 (0.34) BACE1APPMAPT
SCHEMBL3143008 0.88 CHRNB4 (0.39) CHRNB4CHRNA3CHRNA7BACE1MAP4K4
Hydrochloric Acid SCHEMBL3781375 0.88 ABL1 (0.34) BACE1APPMAPT
SCHEMBL3145347 0.87 DHFR (0.37) BACE1APP
Hydrochloric Acid SCHEMBL3773488 0.87 CHRNB4 (0.39) CHRNB4CHRNA3CHRNA7BACE1MAP4K4
SCHEMBL3142890 0.86 KDM1A (0.39) CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL3773421 0.86 DHFR (0.36)
Hydrochloric Acid SCHEMBL3145977 0.85 KDM1A (0.38) CHRNB4CHRNA3CHRNA7
SCHEMBL3147247 0.83 CHRNB4 (0.42) CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed