SCHEMBL31438533

SCHEMBL31438533

[2H]c1cc(NC(C)=O)nc(F)c1C(=O)CBr

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.40
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
ADORA3 P0DMS8 6/20 0.35
ADORA2A P29274 4/20 0.35
CYP1A2 P05177 1/20 0.34
HSP90AA1 P07900 1/20 0.33
HSP90AB1 P08238 1/20 0.33
RAB9A P51151 1/20 0.33
PTPN1 P18031 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ADORA1 P30542 3/20 0.32
ADORA2B P29275 2/20 0.32
MAPT P10636 1/20 0.32
PTK2 Q05397 1/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
MAP4K4 O95819 1/20 0.31
ABL1 P00519 1/20 0.31
CSNK1A1 P48729 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31438540 0.90 MAPK8 (0.35) MAPK8KDM4ELMNAADORA3ADORA2A
SCHEMBL18153003 0.87 MAPK8 (0.42) MAPK8KDM4ELMNAADORA3ADORA2A
SCHEMBL31438557 0.76 MAPK8 (0.42) MAPK8KDM4ELMNAADORA3ADORA2A
SCHEMBL18153007 0.72 PTK2 (0.44) MAPK8KDM4ELMNAADORA3CYP1A2
SCHEMBL25188090 0.72 APP (0.37) PTPN1MAPT
SCHEMBL31438509 0.72 APP (0.37) PTPN1MAPT
SCHEMBL25189945 0.70 KDM4E (0.42) MAPK8KDM4ELMNAADORA3ADORA2A
SCHEMBL24427232 0.69 AKT1 (0.36) MAPK14
SCHEMBL9297719 0.69 KDM4E (0.66) MAPK8KDM4ELMNAHSP90AA1HSP90AB1
SCHEMBL27398573 0.67 ADORA3 (0.46) MAPK8KDM4ELMNAADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116134035-B 3- (1H-imidazol-2-yl) -2,3,8 a-tetrahydroindol-5 (1H) -one derivatives useful as factor XIA inhibitors 詹森药业有限公司 2025-03-11 CN disclosed