SCHEMBL3145508

SCHEMBL3145508

CN(C(=O)O)C1(COc2cnc(Cl)c(-c3ccc(NC(=O)CCl)cc3)c2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
RAB9A P51151 1/20 0.38
GSTO1 P78417 5/20 0.38
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
RNF4 P78317 1/20 0.36
MAP2K7 O14733 2/20 0.36
MALT1 Q9UDY8 3/20 0.35
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3146681 0.86 CHRNB4 (0.45) FFAR4CHRNB4CHRNA3CHRNA7
SCHEMBL3151018 0.85 FFAR4 (0.40) FFAR4CHRNB4CHRNA3CHRNA7
SCHEMBL3147019 0.85 FFAR4 (0.44) FFAR4CHRNB4CHRNA3CHRNA7
SCHEMBL3150647 0.84 FFAR4 (0.40) FFAR4CHRNB4CHRNA3CHRNA7
SCHEMBL3257000 0.84 FFAR4 (0.42) FFAR4CHRNB4CHRNA3CHRNA7
SCHEMBL3147054 0.83 FFAR4 (0.38) FFAR4CHRNB4CHRNA3CHRNA7
Hydrochloric Acid SCHEMBL3778862 0.82 MAP2K7 (0.39) ALDH1A1HTTSMN1; SMN2NPC1MITF
SCHEMBL3773722 0.81 GSTO1 (0.35) ALDH1A1HTTSMN1; SMN2NPC1MITF
SCHEMBL3151256 0.81 FFAR4 (0.38) SMN1; SMN2MAPTMEN1KMT2AFFAR4
SCHEMBL3145499 0.80 ALDH1A1 (0.39) ALDH1A1HTTSMN1; SMN2NPC1MITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed