SCHEMBL3145698

SCHEMBL3145698

O=c1ccc2cccc3c2n1CC3CN1CC[CH]CC1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.39
DRD2 P14416 1/20 0.39
SLC2A1 P11166 1/20 0.34
KCNH2 Q12809 1/20 0.33
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3149594 0.85 HTR1A (0.37) HTR1ADRD2SLC2A1KCNH2CDK4
Hydrochloric Acid SCHEMBL3145852 0.84 HTR1A (0.37) HTR1ADRD2SLC2A1KCNH2CDK4
SCHEMBL3141765 0.79 SLC2A1 (0.42) SLC2A1KCNH2
SCHEMBL3641658 0.79 HTR1A (0.35) HTR1ADRD2
SCHEMBL3394012 0.79 SLC2A1 (0.46) HTR1ADRD2SLC2A1KCNH2
SCHEMBL3676325 0.79 SLC2A1 (0.36) HTR1ADRD2SLC2A1KCNH2
SCHEMBL2291274 0.78 HTR1A (0.43) HTR1ADRD2KCNH2CDK4CCND1
SCHEMBL3209025 0.78 SLC2A1 (0.40) HTR1ADRD2SLC2A1KCNH2
SCHEMBL2287760 0.73 HTR1A (0.40) HTR1ADRD2CDK4CCND1
SCHEMBL3141859 0.72 KCNH2 (0.69) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2136807-B1 PYRROLO (3, 2, 1-IJ) QUINOLINE-4-ONE DERIVATIVES FOR TREATING TUBERCULOSIS GLAXO GROUP LTD (GB) 2010-11-03 EP disclosed
EP-1954697-B1 PERI CONDENSED TRICYCLIC COMPOUNDS USEFUL AS ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2010-02-24 EP disclosed