SCHEMBL31468765

SCHEMBL31468765

Nc1ccc2c(c1)COc1cnccc1-2

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 7/20 0.53
ROCK2 O75116 12/20 0.50
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 1/20 0.50
ROCK1 Q13464 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15972966 0.88 ROCK2 (0.59) AAK1ROCK2
SCHEMBL31468763 0.81 ROCK2 (0.50) AAK1ROCK2ROCK1
SCHEMBL19946104 0.81 ROCK2 (0.56) AAK1ROCK2
SCHEMBL18901287 0.81 AAK1 (0.53) AAK1ROCK2ROCK1
SCHEMBL31474211 0.80 AAK1 (0.49) AAK1ROCK2ROCK1
SCHEMBL31474174 0.79 AAK1 (0.43) AAK1ROCK2LMNAMAPTROCK1
SCHEMBL11558683 0.78 ROCK2 (0.49) AAK1ROCK2ROCK1
SCHEMBL16345579 0.77 ROCK2 (0.69) ROCK2ROCK1
SCHEMBL31468772 0.76 ROCK2 (0.55) AAK1ROCK2LMNAMAPTROCK1
SCHEMBL9671869 0.75 LMNA (0.56) AAK1ROCK2LMNAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025060978-A1 TRICYCLIC PYRIDINE COMPOUND ACTING AS SARM1 ENZYME ACTIVITY INHIBITOR, AND USE THEREOF 科辉智药(深圳)新药研究中心有限公司 2025-03-27 WO disclosed
CN-119661547-A Tricyclic pyridine compounds as SARM1 enzyme activity inhibitors and application thereof 科辉智药(深圳)新药研究中心有限公司 2025-03-21 CN disclosed