SCHEMBL3147249

SCHEMBL3147249

CN(CC1(N(C)C(=O)O)CC1)c1cncc(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.36
SMN1; SMN2 Q16637 5/20 0.36
RAB9A P51151 3/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 2/20 0.36
POLB P06746 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 2/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALOX15 P16050 1/20 0.33
CYP11B2 P19099 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3154940 0.85 SMN1; SMN2 (0.39) HTTSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL3772248 0.83 NPC1 (0.32) HTTSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL3141927 0.79 CYP11B1 (0.32) HTTALDH1A1CYP11B2
SCHEMBL3147244 0.77 HTT (0.35) HTTSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL3772246 0.77 NPC1 (0.33) HTTSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL4820601 0.76 OXTR (0.31)
SCHEMBL3151484 0.75 CHRNB2 (0.38)
SCHEMBL3145942 0.75 HTT (0.38) HTTSMN1; SMN2RAB9AMAPTNPC1
SCHEMBL3776471 0.72 PDE3B (0.36) KDM4EALDH1A1CYP11B2
SCHEMBL4823642 0.72 IDO1 (0.34) SMN1; SMN2POLBTSHRKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed