SCHEMBL3149078

SCHEMBL3149078

Cc1cnn(-c2ccccn2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALKBH2 Q6NS38 1/20 0.57
EGLN1 Q9GZT9 1/20 0.57
GRM4 Q14833 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ALDH1A1 P00352 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
GRM5 P41594 1/20 0.48
DRD2 P14416 2/20 0.46
DRD4 P21917 2/20 0.46
DRD3 P35462 2/20 0.46
MAPT P10636 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP1A2 P05177 2/20 0.44
MTOR P42345 1/20 0.42
MEN1 O00255 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4895758 0.79 KDM4E (0.49) ALKBH2EGLN1SMN1; SMN2ALDH1A1NPC1
SCHEMBL30796754 0.78 GRM5 (0.66) ALKBH2EGLN1GRM4SMN1; SMN2ALDH1A1
SCHEMBL3918642 0.78 GRM5 (0.66) ALKBH2EGLN1GRM4SMN1; SMN2ALDH1A1
SCHEMBL16547471 0.78 ALDH1A1 (0.49) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL5668701 0.78 ALKBH2 (0.57) ALKBH2EGLN1GRM4SMN1; SMN2RAB9A
SCHEMBL2159890 0.78 ALKBH2 (0.57) ALKBH2EGLN1GRM4SMN1; SMN2NPC1
SCHEMBL3923413 0.78 ALKBH2 (0.57) ALKBH2EGLN1GRM4SMN1; SMN2GRM5
SCHEMBL15671484 0.78 EGLN1 (0.57) ALKBH2EGLN1GRM4SMN1; SMN2GRM5
SCHEMBL20658802 0.78 ALKBH2 (0.57) ALKBH2EGLN1GRM4SMN1; SMN2ALDH1A1
SCHEMBL23872054 0.77 ALKBH2 (0.53) ALKBH2EGLN1GRM4SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024044757-A1 AMINOPYRIMIDINE AND AMINOTRIAZINE DERIVATIVES AS MYC PROTEIN MODULATORS Sanford Burnham Prebys Medical Discovery Institute (US) 2024-02-29 WO disclosed
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed
US-11771738-B2 Endoparasitic depsipeptides ZOETIS SERVICES LLC (US) 2023-10-03 US disclosed
US-11771738-B2 Endoparasitic depsipeptides ZOETIS SERVICES LLC (US) 2023-10-03 US disclosed
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
EP-3538519-B1 INDAZOLE DERIVATIVES AS ALPHA V INTEGRIN ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2021-07-28 EP disclosed
EP-3538528-B1 PYRROLE AMIDES AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2020-12-23 EP disclosed
EP-3204360-B1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH INC (US) 2020-08-26 EP disclosed
EP-3209664-B1 BICYCLIC HETEROARYL AMINE COMPOUNDS AS PI3K INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2020-06-03 EP disclosed
EP-0846113-B1 1-(PYRIDYL)-PYRAZOLS AND THEIR USE AS HERBICIDES BASF AG (DE) 2003-01-29 EP disclosed
EP-0759429-B1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF AG (DE) 2001-10-24 EP disclosed
EP-0846113-A1 1-(PYRIDYL)-PYRAZOLS AND THEIR USE AS HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1998-06-10 EP disclosed
WO-1997007114-A1 1-(PYRIDYL)-PYRAZOLS AND THEIR USE AS HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1997-02-27 WO disclosed
EP-0759429-A1 Substituted trifluormethylpyridines useful as intermediates for herbicidal 1-(pyridyl)-pyrazoles BASF Aktiengesellschaft (DE) 1997-02-26 EP disclosed
EP-0366329-B1 Halogeno-4-methylpyrazoles and process for preparing the same NISSAN CHEMICAL IND LTD (JP) 1996-03-20 EP disclosed
US-5220028-A Halogeno-4-methylpyrazoles NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1993-06-15 US disclosed
EP-0366328-B1 PROCESS FOR PREPARING 4-METHYLPYRAZOLES NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1993-05-19 EP disclosed
EP-0366329-A1 Halogeno-4-methylpyrazoles and process for preparing the same NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1990-05-02 EP disclosed
EP-0366328-A1 Process for preparing 4-methylpyrazoles NISSAN CHEMICAL INDUSTRIES, LIMITED (JP) 1990-05-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11771738-B2 Endoparasitic depsipeptides VIP, PREP, VIPR1 ALKBH2 4823/4885EGLN1 239/4885GRM4 2485/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.