SCHEMBL3149462

SCHEMBL3149462

COc1ccccc1-c1ccc2nc[nH]c2c1CN

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.57
DPP8 Q6V1X1 2/20 0.40
LRRK2 Q5S007 2/20 0.39
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38
ABL1 P00519 1/20 0.38
RAD52 P43351 1/20 0.38
RIN1 Q13671 1/20 0.38
ALDH1A1 P00352 1/20 0.38
IDO1 P14902 1/20 0.38
METAP2 P50579 1/20 0.38
HTR7 P34969 1/20 0.38
HTR3A P46098 1/20 0.37
MAP4K4 O95819 1/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37
CCNB2 O95067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3149686 0.77 DPP4 (0.60) DPP4DPP8SMN1; SMN2
SCHEMBL3143679 0.73 DPP4 (1.00) DPP4DPP8
SCHEMBL1993654 0.71 DPP4 (0.45) DPP4ALDH1A1SMN1; SMN2
SCHEMBL3149112 0.71 DPP4 (0.45) DPP4ALDH1A1SMN1; SMN2HSD17B10
SCHEMBL8277153 0.70 DPP4 (0.64) DPP4DPP8
SCHEMBL3082549 0.70 ABL1 (0.54) ABL1RAD52RIN1ALDH1A1TP53
SCHEMBL31538912 0.69 ABL1 (0.53) ABL1RAD52RIN1ALDH1A1TP53
SCHEMBL5158690 0.67 DPP4 (0.46) DPP4ALDH1A1HSD17B10GSK3B
SCHEMBL1996958 0.67 DPP4 (0.46) DPP4LRRK2ALDH1A1HTR7HSD17B10
SCHEMBL7345542 0.66 ABL1 (0.45) ABL1RAD52RIN1SMN1; SMN2CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687638-B2 Dipeptidyl peptidase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-03-30 US disclosed
US-7687638-B2 Dipeptidyl peptidase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-03-30 US disclosed
US-7687638-B2 Dipeptidyl peptidase inhibitors TAKEDA SAN DIEGO, INC. (US) 2010-03-30 US disclosed
WO-2005118555-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-12-15 WO disclosed