SCHEMBL5158690

SCHEMBL5158690

COc1ccccc1-c1ccc2c(c1CN)[N]C(=O)N2

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.46
CHEK1 O14757 1/20 0.39
HSD17B10 Q99714 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
KDM4E B2RXH2 2/20 0.37
GPR55 Q9Y2T6 1/20 0.37
AR P10275 1/20 0.36
CREBBP Q92793 1/20 0.36
STK10 O94804 2/20 0.36
SLK Q9H2G2 2/20 0.36
PTPRC P08575 1/20 0.35
PTPN1 P18031 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
C1R P00736 1/20 0.34
GSK3B P49841 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5325810 0.88 DPP4 (0.45) DPP4CHEK1HSD17B10ALDH1A1GAA
SCHEMBL1996958 0.70 DPP4 (0.46) DPP4HSD17B10ALDH1A1GAAKDM4E
SCHEMBL1993654 0.69 DPP4 (0.45) DPP4CHEK1ALDH1A1KDM4EPTPRC
SCHEMBL3149112 0.69 DPP4 (0.45) DPP4CHEK1HSD17B10ALDH1A1GAA
SCHEMBL3149462 0.67 DPP4 (0.57) DPP4HSD17B10ALDH1A1GSK3B
SCHEMBL6867119 0.66 TAAR1 (0.55) DPP4HSD17B10ALDH1A1GAA
SCHEMBL4139350 0.63 IL6 (0.39) CHEK1HSD17B10ALDH1A1GAAKDM4E
SCHEMBL23611757 0.63 HSD17B10 (0.66) HSD17B10ALDH1A1GAAKDM4EGSK3B
SCHEMBL3143679 0.63 DPP4 (1.00) DPP4
SCHEMBL301996 0.63 CA1 (0.71) HSD17B10ALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1753730-A1 DIPEPTIDYL PEPTIDASE INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2007-02-21 EP claimed
WO-2005118555-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-12-15 WO claimed
EP-1753730-A1 DIPEPTIDYL PEPTIDASE INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2007-02-21 EP disclosed
WO-2005118555-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-12-15 WO disclosed