SCHEMBL3149710

SCHEMBL3149710

Cc1cc(OCc2c(C(C)C)nnn2-c2ccccc2OC(F)(F)F)ccc1-c1ccc(C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.46
HSD17B13 Q7Z5P4 1/20 0.39
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
PPARD Q03181 8/20 0.37
PPARA Q07869 4/20 0.36
PPARG P37231 2/20 0.36
CETP P11597 1/20 0.36
KCNH2 Q12809 1/20 0.36
TRPM8 Q7Z2W7 2/20 0.36
NTRK1 P04629 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27761419 0.92 NR1H4 (0.38) NR1H4PPARDPPARAPPARGNTRK1
SCHEMBL3165823 0.92 NR1H4 (0.51) NR1H4HSD17B13RXRARXRBRXRG
SCHEMBL3158844 0.89 NR1H4 (0.47) NR1H4RXRARXRBRXRGPPARD
SCHEMBL3159951 0.86 NR1H4 (0.46) NR1H4HSD17B13RXRARXRBRXRG
SCHEMBL2770877 0.86 NR1H4 (0.42) NR1H4HSD17B13RXRARXRBRXRG
SCHEMBL3156107 0.86 NR1H4 (0.39) NR1H4PPARDPPARA
SCHEMBL3150730 0.85 NR1H4 (0.41) NR1H4PPARDPPARAPPARGFFAR4
SCHEMBL3159296 0.83 NR1H4 (0.61) NR1H4
SCHEMBL3159291 0.83 NR1H4 (0.61) NR1H4
SCHEMBL498384 0.82 NR1H4 (0.44) NR1H4PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029558-B1 COMPOUNDS AND METHODS FOR MODULATING FXR LILLY CO ELI (US) 2010-03-10 EP disclosed