SCHEMBL3157696

SCHEMBL3157696

O=C(c1ccc(S(=O)(=O)Nc2ccccc2Oc2ccc(Cl)cc2Cl)cc1)N1CCN(CCCN2CCCCC2)CC1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 9/20 0.51
L3MBTL1 Q9Y468 1/20 0.47
KCNH2 Q12809 1/20 0.47
RXFP1 Q9HBX9 1/20 0.45
CCR1 P32246 1/20 0.45
HRH3 Q9Y5N1 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3153878 0.99 CCR2 (0.50) CCR2L3MBTL1KCNH2RXFP1CCR1
SCHEMBL3148147 0.98 CCR2 (0.49) CCR2L3MBTL1KCNH2RXFP1KMT2A
SCHEMBL3148887 0.97 CCR2 (0.53) CCR2L3MBTL1KCNH2RXFP1CCR1
SCHEMBL3149703 0.96 CCR2 (0.51) CCR2L3MBTL1KCNH2RXFP1CCR1
SCHEMBL3148157 0.92 GAA (0.46) CCR2L3MBTL1RXFP1KMT2A
SCHEMBL3154679 0.92 GAA (0.49) CCR2L3MBTL1CCR1KMT2A
SCHEMBL3158340 0.90 CACNA1H (0.44) CCR2L3MBTL1CCR1KMT2A
SCHEMBL3145106 0.89 F10 (0.49) CCR2L3MBTL1RXFP1CCR1KMT2A
SCHEMBL3148378 0.89 GAA (0.49) CCR2L3MBTL1CCR1KMT2A
SCHEMBL3273918 0.89 CCR2 (0.55) CCR2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074083-B1 NEW SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS RICHTER GEDEON NYRT (HU) 2013-06-19 EP disclosed
US-20100075978-A1 SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS RICHTER GEDEON NYRT. (HU) 2010-03-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100075978-A1 SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS BDKRB1, BDKRB2, TRPV1 CCR2 417/4885L3MBTL1 3132/4885KCNH2 80/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.