SCHEMBL316068

SCHEMBL316068

Cc1onc(-c2ccccc2Cl)c1C(=O)NC1CCC(Cc2cccc(F)c2)(N(C)C)CC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.60
GPBAR1 Q8TDU6 2/20 0.53
MAPT P10636 1/20 0.50
GHSR Q92847 1/20 0.49
MEN1 O00255 2/20 0.49
ALDH1A1 P00352 3/20 0.48
TSHR P16473 1/20 0.48
LMNA P02545 3/20 0.48
HTT P42858 1/20 0.48
CYP2C19 P33261 1/20 0.47
EPAS1 Q99814 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316443 0.93 GHSR (0.58) KMT2AMAPTGHSRMEN1ALDH1A1
SCHEMBL316325 0.92 KMT2A (0.61) KMT2AGPBAR1MAPTGHSRMEN1
SCHEMBL316534 0.91 KMT2A (0.58) KMT2AMAPTGHSRMEN1ALDH1A1
SCHEMBL315598 0.91 KMT2A (0.62) KMT2AGPBAR1MAPTGHSRMEN1
SCHEMBL315482 0.86 KMT2A (0.62) KMT2AGPBAR1MAPTGHSRMEN1
SCHEMBL316299 0.85 KMT2A (0.57) KMT2AMAPTGHSRMEN1ALDH1A1
SCHEMBL314979 0.85 GHSR (0.62) KMT2AMAPTGHSRMEN1ALDH1A1
SCHEMBL316457 0.85 GHSR (0.54) KMT2AGPBAR1MAPTGHSRMEN1
SCHEMBL315615 0.85 KMT2A (0.62) KMT2AGPBAR1MAPTGHSRALDH1A1
SCHEMBL315886 0.84 GHSR (0.60) KMT2AMAPTGHSRMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed