SCHEMBL315482

SCHEMBL315482

Cc1onc(-c2ccccc2Cl)c1C(=O)NC1CCC(Cc2ccccc2F)(N(C)C)CC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.62
GPBAR1 Q8TDU6 1/20 0.51
ALDH1A1 P00352 3/20 0.50
TSHR P16473 1/20 0.50
GHSR Q92847 2/20 0.49
CYP2C19 P33261 2/20 0.48
LMNA P02545 2/20 0.48
NPC1 O15118 1/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 1/20 0.48
MEN1 O00255 1/20 0.47
CYP3A4 P08684 1/20 0.47
RECQL P46063 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316102 0.92 GHSR (0.56) KMT2AALDH1A1GHSRLMNANPC1
SCHEMBL315545 0.92 GHSR (0.59) KMT2AALDH1A1GHSRLMNANPC1
SCHEMBL316058 0.92 KMT2A (0.65) KMT2AGPBAR1ALDH1A1TSHRGHSR
SCHEMBL315598 0.88 KMT2A (0.62) KMT2AGPBAR1ALDH1A1TSHRGHSR
SCHEMBL316040 0.88 GHSR (0.55) KMT2AALDH1A1GHSRLMNANPC1
SCHEMBL316068 0.86 KMT2A (0.60) KMT2AGPBAR1ALDH1A1TSHRGHSR
SCHEMBL316283 0.85 GHSR (0.62) KMT2AALDH1A1TSHRGHSRMAPT
SCHEMBL316325 0.84 KMT2A (0.61) KMT2AGPBAR1ALDH1A1TSHRGHSR
SCHEMBL316299 0.84 KMT2A (0.57) KMT2AALDH1A1GHSRLMNANPC1
SCHEMBL315424 0.84 GHSR (0.61) KMT2AALDH1A1TSHRGHSRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed