SCHEMBL3169166

SCHEMBL3169166

CC(=O)NCCNc1cc(NCCNC(=O)Cc2ccc(-c3ccccc3)cc2)nc(-c2ccc(Cl)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
ADAMTS5 Q9UNA0 1/20 0.45
KMT2A Q03164 5/20 0.44
CYP3A4 P08684 3/20 0.44
HPGD P15428 3/20 0.44
MEN1 O00255 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
PDE4B Q07343 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ADORA3 P0DMS8 2/20 0.44
LTA4H P09960 1/20 0.43
EPHX2 P34913 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
LMNA P02545 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3170639 0.96 KMT2A (0.48) ALDH1A1SMN1; SMN2CNR1CNR2KMT2A
SCHEMBL3162245 0.95 ALDH1A1 (0.47) ALDH1A1KMT2ACYP3A4MEN1CYP1A2
SCHEMBL3164379 0.91 TP53 (0.52) ALDH1A1SMN1; SMN2CNR2KMT2AHPGD
SCHEMBL3156387 0.90 ADORA2A (0.48) ALDH1A1CYP3A4HPGDCYP1A2CYP2D6
SCHEMBL3177073 0.90 CYP1A2 (0.47) ALDH1A1SMN1; SMN2KMT2AMEN1CYP1A2
SCHEMBL3171179 0.89 KMT2A (0.50) ALDH1A1KMT2ACYP3A4HPGDMEN1
SCHEMBL3176265 0.88 MEN1 (0.50) SMN1; SMN2CNR2KMT2AMEN1ADORA3
SCHEMBL3166463 0.88 CNR1 (0.47) ALDH1A1CNR1CNR2CYP3A4CYP1A2
SCHEMBL3172697 0.86 NPC1 (0.47) ALDH1A1SMN1; SMN2KMT2ACYP3A4MEN1
SCHEMBL3163028 0.86 KMT2A (0.47) ALDH1A1SMN1; SMN2CNR1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465631-B1 PYRIMIDINE A2B SELECTIVE ANTAGONIST COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2010-02-24 EP disclosed