SCHEMBL3176265

SCHEMBL3176265

COc1ccc(CC(=O)NCCNc2cc(NCCNC(C)=O)nc(-c3ccc(Cl)cc3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
TP53 P04637 3/20 0.50
CLK4 Q9HAZ1 1/20 0.47
SCD O00767 1/20 0.46
ADORA3 P0DMS8 2/20 0.46
CNR2 P34972 1/20 0.46
KDR P35968 2/20 0.46
CSNK1D P48730 1/20 0.46
THRB P10828 1/20 0.45
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
PTGDR Q13258 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
ADORA2B P29275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3166238 0.90 ALDH1A1 (0.54) CLK4ADORA3THRBPTGDRSMN1; SMN2
SCHEMBL3171330 0.90 CA1 (0.48) TP53CLK4SMN1; SMN2
SCHEMBL3164379 0.89 TP53 (0.52) MEN1KMT2ATP53ADORA3CNR2
SCHEMBL3169166 0.88 ALDH1A1 (0.49) MEN1KMT2ATP53ADORA3CNR2
SCHEMBL3177073 0.88 CYP1A2 (0.47) MEN1KMT2ATP53ADORA3THRB
SCHEMBL3170639 0.88 KMT2A (0.48) MEN1KMT2ATP53CLK4ADORA3
SCHEMBL3171746 0.87 TP53 (0.49) MEN1KMT2ATP53CLK4SCD
SCHEMBL3170716 0.87 MAPT (0.53) MEN1KMT2ATP53CLK4SCD
SCHEMBL3170868 0.87 LMNA (0.49) TP53ADORA3KDR
SCHEMBL3177128 0.87 LMNA (0.49) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465631-B1 PYRIMIDINE A2B SELECTIVE ANTAGONIST COMPOUNDS, THEIR SYNTHESIS AND USE OSI PHARM INC (US) 2010-02-24 EP disclosed