SCHEMBL3171972

SCHEMBL3171972

NC(=O)c1nc2c(s1)CCCC2C(=O)N1CCN(c2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
TFPI2 P48307 1/20 0.43
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
RECQL P46063 2/20 0.43
POLB P06746 1/20 0.43
NR4A1 P22736 1/20 0.43
BLM P54132 1/20 0.43
ESR2 Q92731 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ADAM10 O14672 1/20 0.42
ERBB2 P04626 1/20 0.42
MMP2 P08253 1/20 0.42
TP53 P04637 2/20 0.41
NPSR1 Q6W5P4 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175350 0.91 LSS (0.39) ALDH1A1SMN1; SMN2MAPTMAPK1HTT
SCHEMBL3156915 0.88 MAPT (0.51) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL3171977 0.87 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2MAPTMAPK1HTT
SCHEMBL3170296 0.86 SMN1; SMN2 (0.43) ALDH1A1SMN1; SMN2MAPTMAPK1KMT2A
SCHEMBL3163988 0.86 KDM4E (0.48) ALDH1A1SMN1; SMN2MAPTMAPK1HTT
SCHEMBL3157437 0.85 GRM5 (0.41) ALDH1A1SMN1; SMN2HTTRECQLTSHR
SCHEMBL3157536 0.83 CHRM3 (0.43) ALDH1A1KMT2AMEN1BLMNPSR1
SCHEMBL3167878 0.82 POLB (0.38) MAPTHTTTFPI2POLBL3MBTL1
SCHEMBL3165721 0.80 DHODH (0.43) ALDH1A1HTTKMT2AMEN1POLB
SCHEMBL3175358 0.78 CHRM1 (0.40) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716128-B1 SUBSTITUTED 4,5,6,7-TETRAHYDRO-BENZOTHIAZOL-2-YLAMINE COMPOUNDS GRUENENTHAL GMBH (DE) 2010-03-31 EP claimed