SCHEMBL31745274

SCHEMBL31745274

Clc1ccc2nccc(Br)c2n1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.40
RPS6KA5 O75582 1/20 0.33
RPS6KA4 O75676 1/20 0.33
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
NR4A2 P43354 1/20 0.32
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
NQO2 P16083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15884328 0.79 NQO2 (0.34) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL23147517 0.79 CRHBP (0.36) EGFRRPS6KA5RPS6KA4NR4A2CRHBP
SCHEMBL29582669 0.76 EGFR (0.40) EGFRADRA2AADRA2BADRA2CADRA1D
SCHEMBL796213 0.76 ACHE (0.39) EGFRRPS6KA5RPS6KA4ADRA1ANR4A2
SCHEMBL22715644 0.76 NR4A2 (0.47) EGFRRPS6KA5RPS6KA4NR4A2
SCHEMBL24422788 0.76 EGFR (0.40) EGFRADRA2AADRA2BADRA2CADRA1D
SCHEMBL15884240 0.76 NQO2 (0.36) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL29472071 0.76 ACHE (0.39) EGFRRPS6KA5RPS6KA4ADRA1ANR4A2
SCHEMBL14905208 0.74 EGFR (0.39) EGFR
SCHEMBL14905211 0.72 EGFR (0.38) EGFRADRA2AADRA2BADRA2CNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250382301-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF UNIV ARIZONA (US) 2025-12-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250382301-A1 SMALL MOLECULE INHIBITORS OF DYRK/CLK AND USES THEREOF CLK2, CLK3, CLK1 EGFR 592/4885RPS6KA5 125/4885RPS6KA4 218/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.