SCHEMBL3177399

SCHEMBL3177399

CC(C)(N)n1ccc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.42
CCND1 P24385 4/20 0.42
NOTUM Q6P988 1/20 0.41
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR6 P50406 1/20 0.37
BIRC5 O15392 1/20 0.36
LMNA P02545 1/20 0.36
CA12 O43570 2/20 0.35
CA9 Q16790 2/20 0.35
BRD4 O60885 1/20 0.35
BRPF1 P55201 1/20 0.35
KAT2B Q92831 1/20 0.35
BRD9 Q9H8M2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL645711 0.83 CDK4 (0.45) CDK4CCND1NOTUMHTR2AHTR2C
SCHEMBL24218236 0.79 CDK4 (0.42) CDK4CCND1NOTUMHTR2AHTR2C
SCHEMBL1724156 0.79 CDK4 (0.42) CDK4CCND1NOTUMHTR2AHTR2C
SCHEMBL12386866 0.76 CDK4 (0.44) CDK4CCND1NOTUMHTR2AHTR2C
Bicarbonate SCHEMBL28410218 0.75 NOTUM (0.50) CDK4CCND1NOTUMHTR6LMNA
SCHEMBL16719593 0.75
SCHEMBL22549893 0.74 CDK4 (0.45) CDK4CCND1NOTUMHTR6BIRC5
SCHEMBL31066760 0.74 CDK4 (0.45) CDK4CCND1NOTUMHTR2AHTR2C
SCHEMBL30144 0.74 CDK4 (0.45) CDK4CCND1NOTUMHTR2AHTR2C
SCHEMBL19996599 0.73 CDK4 (0.38) CDK4CCND1NOTUMHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8410075-B2 Mannich base N-oxide drugs CASCADE PRODRUG INC. (US) 2013-04-02 US disclosed
US-20100016252-A1 Mannich Base N-Oxide Drugs State of Oregon Acting By and Through The Oregon State Board of Higher Education On Behalf of The U (US) 2010-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016252-A1 Mannich Base N-Oxide Drugs ASAH2, MAN2B1, NNT CDK4 2781/4885CCND1 4181/4885NOTUM 2521/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.