SCHEMBL3198709

SCHEMBL3198709

CC1(C)CN(c2c(F)cc3c(=O)c(C(=O)O)cn([C@@H]4C[C@H]4F)c3c2Cl)CC1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
POLB P06746 3/20 0.60
OPRM1 P35372 2/20 0.60
CHRM2 P08172 1/20 0.60
CHRM1 P11229 1/20 0.60
OPRD1 P41143 1/20 0.60
CYP3A4 P08684 2/20 0.48
CYP2C9 P11712 1/20 0.48
KCNH2 Q12809 5/20 0.45
AADAT Q8N5Z0 2/20 0.42
KDM4E B2RXH2 5/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.41
TOP1 P11387 2/20 0.41
HPGD P15428 3/20 0.41
HSD17B10 Q99714 3/20 0.41
ALB P02768 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3198715 1.00 ALDH1A1 (0.60) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL8509346 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL29821427 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL2784482 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL29368438 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL74553 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL13483604 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL1652843 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL21416358 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
Sitafloxacin Anhydrous SCHEMBL3198924 0.90 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE41149-E1 Stereoisomerically pure 7-[(7S)-7-amino-5-azaspiro[2.4]heptan-5-yl]-6-fluoro-1-[(1R,2S)-2-fluoro-1-cyclopropyl]-8-methoxy-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid or a pharmaceutically acceptable salt thereof; antibacterial agents DAIICHI SANKYO COMPANY, LIMITED (JP) 2010-02-23 US disclosed
US-6031102-A Optically active pyridonecarboxylic acid derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2000-02-29 US disclosed
US-5587386-A BACTERICIDES, MICROBIOCIDES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed