SCHEMBL3203395

SCHEMBL3203395

C1=CN=Cc2cc3ccccc3n2C1

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.35
HTR2C P28335 5/20 0.35
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1864062 0.77 HTR2A (0.40) HTR2AHTR2CNOTUM
SCHEMBL29851785 0.77 HTR2A (0.40) HTR2AHTR2CNOTUM
SCHEMBL3211491 0.72 HTR2A (0.37) HTR2AHTR2CNOTUM
Hydroxyamine SCHEMBL9656520 0.72 HTR2A (0.37) HTR2AHTR2CNOTUM
SCHEMBL4017486 0.72 HTR2A (0.39) HTR2AHTR2CNOTUM
SCHEMBL29538429 0.72 HTR2A (0.39) HTR2AHTR2CNOTUM
SCHEMBL30864980 0.69 HTR2A (0.40) HTR2AHTR2CNOTUM
SCHEMBL5253279 0.65 DAO (0.40)
SCHEMBL18229897 0.65 HTR2A (0.49) HTR2AHTR2CNOTUM
SCHEMBL4860771 0.63 HTR2A (0.30) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790712-B2 Substituted [1,4]diazepino[1,2-A]indoles and azepino[1,2-A]indoles as anti-cytokine inhibitors BOEHRINGER INGELHEIM PHARMACEUTICAL, INC. (US) 2010-09-07 US disclosed