SCHEMBL321513

SCHEMBL321513

Nc1[nH]ncc1-c1cc(-c2ccc(C(F)(F)F)cc2)ccc1Oc1cc(F)c(S(=O)(=O)Nc2cscn2)cc1Cl

nearest known ligand 0.89

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 20/20 0.89
CYP2C9 P11712 4/20 0.89
SCN5A Q14524 4/20 0.89
SCN2B O60939 1/20 0.78
SCN1A P35498 1/20 0.78
SCN4A P35499 1/20 0.78
SCN7A Q01118 1/20 0.78
SCN1B Q07699 1/20 0.78
SLC22A12 Q96S37 1/20 0.78
SCN2A Q99250 1/20 0.78
SCN3A Q9NY46 1/20 0.78
SCN8A Q9UQD0 1/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17450366 0.94 SCN9A (1.00) SCN9ACYP2C9SCN5ASCN2BSCN1A
Pf-05089771 SCHEMBL1095065 0.88 SCN9A (1.00) SCN9ACYP2C9SCN5ASCN2BSCN1A
Pf-05089771 SCHEMBL31060533 0.88 SCN9A (1.00) SCN9ACYP2C9SCN5ASCN2BSCN1A
Pf-05089771 SCHEMBL29376793 0.88 SCN9A (1.00) SCN9ACYP2C9SCN5ASCN2BSCN1A
SCHEMBL319970 0.88 SCN9A (0.88) SCN9ACYP2C9SCN5ASCN2BSCN1A
Trifluoroacetic Acid SCHEMBL14889980 0.85 SCN9A (0.79) SCN9ACYP2C9SCN5ASCN2BSCN1A
SCHEMBL1690669 0.85 SCN9A (0.90) SCN9ACYP2C9SCN5ASCN1ASCN2A
SCHEMBL31643102 0.82 SCN9A (0.78) SCN9ACYP2C9SCN5ASCN2BSCN1A
SCHEMBL1094748 0.82 SCN9A (0.78) SCN9ACYP2C9SCN5ASCN2BSCN1A
SCHEMBL16531374 0.82 SCN9A (1.00) SCN9ACYP2C9SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590951-B1 BENZENESULFONAMIDES USEFUL AS SODIUM CHANNEL INHIBITORS PFIZER LTD (GB) 2015-01-07 EP disclosed
US-8772293-B2 Chemical compounds PFIZER LIMITED (GB) 2014-07-08 US disclosed
EP-2590951-A1 BENZENESULFONAMIDES USEFUL AS SODIUM CHANNEL INHIBITORS Pfizer Limited (GB) 2013-05-15 EP disclosed
WO-2012004743-A1 BENZENESULFONAMIDES USEFUL AS SODIUM CHANNEL INHIBITORS PFIZER LIMITED (GB) 2012-01-12 WO disclosed
US-20120010182-A1 Chemical Compounds ICAGEN INC. (US) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010182-A1 Chemical Compounds SCN1A, SCN1B, CACNA1E SCN9A 12/4885CYP2C9 533/4885SCN5A 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.