SCHEMBL3218445

SCHEMBL3218445

O=C1N=c2cc(Cl)c(Cl)c(Cl)c2=N1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
AHR P35869 1/20 0.30
HPGD P15428 2/20 0.30
TSHR P16473 2/20 0.30
HSD17B10 Q99714 2/20 0.30
HSP90AA1 P07900 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362276 0.82 ALDH1A1 (0.33) CYP3A4
SCHEMBL3223624 0.77
SCHEMBL6908764 0.76 GRIN2D (0.31) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL3539564 0.76 KDM4E (0.36) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL6839545 0.74 AHR (0.33) CYP3A4AHRMAPK1
SCHEMBL3226843 0.74 ALDH1A1 (0.35) CYP3A4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL11657600 0.71 KDM4E (0.31)
SCHEMBL7491378 0.71 GRIN2D (0.33) CYP3A4GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7498714 0.71 CYP3A4 (0.39) CYP3A4TSHR
SCHEMBL1115538 0.67 GAA (0.48) CYP3A4HPGDTSHRHSD17B10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015037-A1 THERAPEUTIC METHODS AND COMPOSITIONS HOWARD FLOREY INSTITUTE (AU) 2010-02-11 WO disclosed