SCHEMBL321895

SCHEMBL321895

CNC(=O)/C(=N/OC)c1ccccc1/C=N/OCCc1cccc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.41
ALOX5 P09917 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
TDP1 Q9NUW8 1/20 0.36
RXFP1 Q9HBX9 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
NR1I2 O75469 1/20 0.35
ADRB1 P08588 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL154410 1.00 HIF1A (0.41) HIF1AALOX5SIRT2KDM4EALDH1A1
SCHEMBL15650134 1.00 HIF1A (0.41) HIF1AALOX5SIRT2KDM4EALDH1A1
SCHEMBL8760920 0.91 HIF1A (0.44) HIF1AKDM4EALDH1A1SMN1; SMN2MEN1
SCHEMBL13519408 0.89 HDAC1 (0.34) HIF1AALOX5HDAC1
SCHEMBL13519406 0.89 HDAC1 (0.34) HIF1AALOX5HDAC1
SCHEMBL7870291 0.82 ALOX5 (0.39) HIF1AALOX5SIRT2KDM4EALDH1A1
SCHEMBL8760949 0.81 HIF1A (0.54) HIF1AKDM4EMAPT
SCHEMBL8760953 0.81 HIF1A (0.54) HIF1AKDM4EMAPT
SCHEMBL7178443 0.81 HIF1A (0.42) HIF1AALOX5SIRT2KDM4EALDH1A1
SCHEMBL7876786 0.80 ALOX5 (0.37) HIF1AALOX5SIRT2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 122 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3490379-A1 ACTIVE COMPOUND COMBINATIONS AND METHODS TO PROTECT THE PROPAGATION MATERIAL OF PLANTS Bayer CropScience Aktiengesellschaft (DE) 2019-06-05 EP claimed
WO-2018019676-A1 ACTIVE COMPOUND COMBINATIONS AND METHODS TO PROTECT THE PROPAGATION MATERIAL OF PLANTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2018-02-01 WO claimed
EP-3010893-A1 ARYL SULFIDE DERIVATIVES AND ARYL SULFOXIDE DERIVATIVES AS ACARICIDES AND INSECTICIDES Bayer CropScience Aktiengesellschaft (DE) 2016-04-27 EP claimed
WO-2014202510-A1 ARYL SULFIDE DERIVATIVES AND ARYL SULFOXIDE DERIVATIVES AS ACARICIDES AND INSECTICIDES BAYER CROPSCIENCE AG (DE) 2014-12-24 WO claimed
EP-2651209-A2 SOYBEAN EVENT SYHT0H2 AND COMPOSITIONS AND METHODS FOR DETECTION THEREOF Syngenta Participations AG (CH) 2013-10-23 EP claimed
EP-2597951-A2 USE OF SUCCINATE DEHYDROGENASE INHIBITORS AND/OR RESPIRATORY CHAIN COMPLEX III INHIBITORS FOR IMPROVING THE RATIO OF HARMFUL TO BENEFICIAL MICROORGANISMS Bayer Intellectual Property GmbH (DE) 2013-06-05 EP claimed
EP-2590511-A2 ANTHRANILAMIDES IN COMBINATION WITH FUNGICIDES Bayer Intellectual Property GmbH (DE) 2013-05-15 EP claimed
EP-2477497-A2 SYNERGISTIC FUNGICIDAL COMBINATIONS CONTAINING A DITHIINO-TETRACARBOXAMIDE FUNGICIDE Bayer CropScience AG (DE) 2012-07-25 EP claimed
WO-2012082548-A2 SOYBEAN EVENT SYHT0H2 AND COMPOSITIONS AND METHODS FOR DETECTION THEREOF SYNGENTA PARTICIPATIONS AG (CH) 2012-06-21 WO claimed
EP-2451277-A2 PROCESS FOR IMPROVING SEEDLING GROWTH AND/OR EARLY EMERGENCE OF CROPS Bayer CropScience AG (DE) 2012-05-16 EP claimed
WO-2012013590-A2 USE OF SUCCINATE DEHYDROGENASE INHIBITORS AND/OR RESPIRATORY CHAIN COMPLEX III INHIBITORS FOR IMPROVING THE RATIO OF HARMFUL TO BENEFICIAL MICROORGANISMS BAYER CROPSCIENCE AG (DE) 2012-02-02 WO claimed
WO-2012004221-A2 ANTHRANILAMIDES IN COMBINATION WITH FUNGICIDES BAYER CROPSCIENCE AG (DE) 2012-01-12 WO claimed
WO-2011029551-A2 ACTIVE COMPOUND COMBINATIONS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2011-03-17 WO claimed
WO-2011003533-A2 PROCESS FOR IMPROVING SEEDLING GROWTH AND/OR EARLY EMERGENCE OF CROPS BAYER CROPSCIENCE AG (DE) 2011-01-13 WO claimed
WO-2019150311-A1 1-3 DITHIOL COMPOUNDS AND THEIR USE FOR THE PROTECTION OF CROPS FROM PHYTOPATHOGENIC MICROORGANISMS PI INDUSTRIES LTD. (IN) 2019-08-08 WO disclosed
EP-3481195-A1 AQUEOUS COMPOSITIONS FOR TREATING SEEDS, SEEDS TREATED THEREWITH, AND METHODS FOR TREATING SEEDS Covestro LLC, ET AL. (US) 2019-05-15 EP disclosed
EP-3481194-A1 AQUEOUS COMPOSITIONS FOR TREATING SEEDS, SEEDS TREATED THEREWITH, AND METHODS FOR TREATING SEEDS Covestro LLC, ET AL. (US) 2019-05-15 EP disclosed
WO-2010121735-A1 USE OF PROPINEB AS BIRD REPELLENT BAYER CROPSCIENCE AG (DE) 2010-10-28 WO disclosed
WO-2010094666-A2 FUNGICIDAL N-(PHENYLCYCLOALKYL)CARBOXAMIDE, N-(BENZYLCYCLOALKYL)CARBOXAMIDE AND THIOCARBOXAMIDE DERIVATIVES BAYER CROPSCIENCE AG (DE) 2010-08-26 WO disclosed
WO-2009068194-A2 HALOGEN-SUBSTITUTED Δ1 PYRROLINES BAYER CROPSCIENCE AG (DE) 2009-06-04 WO disclosed