SCHEMBL3225907

SCHEMBL3225907

O=C(O)CC1(c2ccc(Nc3nc(NCCc4ccccc4)cc(-c4ccccc4)n3)cc2)CCC1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.42
HRH4 Q9H3N8 2/20 0.42
VCP P55072 8/20 0.40
SYK P43405 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
BRAF P15056 1/20 0.38
PTGDR Q13258 1/20 0.36
SLC2A1 P11166 1/20 0.36
KCNH3 Q9ULD8 1/20 0.36
HDAC1 Q13547 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
POLB P06746 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3227460 0.87 PTGDR (0.46) HRH1HRH4VCPSYKBRAF
SCHEMBL3232266 0.84 HRH1 (0.45) HRH1HRH4VCPBRAFPTGDR
SCHEMBL3234459 0.81 CAMK2D (0.45) VCPSYKMEN1KMT2A
SCHEMBL3420476 0.81 CAMK2D (0.45) VCPSYKMEN1KMT2A
SCHEMBL3221036 0.77 PTGDR (0.47) HRH4VCPSYKPTGDR
SCHEMBL3225921 0.76 ADORA1 (0.36) VCPSLC2A1MEN1KMT2A
SCHEMBL13456904 0.74 VCP (0.48) HRH1HRH4VCP
SCHEMBL3236008 0.74 PTGDR (0.45) HRH1HRH4VCPSYKPTGDR
SCHEMBL3261619 0.73 VCP (0.42) VCPSYKPTGDR
SCHEMBL3235448 0.72 SYK (0.42) VCPSYKNPC1POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028179-A1 HETEROCYCLIC COMPOUNDS AS GATA MODULATORS DR. REDDY'S LABORATORIES LTD. (IN) 2010-03-11 WO claimed
WO-2010028179-A1 HETEROCYCLIC COMPOUNDS AS GATA MODULATORS DR. REDDY'S LABORATORIES LTD. (IN) 2010-03-11 WO disclosed