SCHEMBL3228522

SCHEMBL3228522

NC(=O)C(CCCCC(=O)Nc1ccccn1)c1ccc(F)cc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 6/20 0.53
HDAC1 Q13547 6/20 0.53
HDAC4 P56524 4/20 0.53
HDAC7 Q8WUI4 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC10 Q969S8 3/20 0.53
HDAC11 Q96DB2 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC9 Q9UKV0 3/20 0.53
HDAC5 Q9UQL6 3/20 0.53
GAA P10253 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MEF2D Q14814 1/20 0.44
NPC1 O15118 3/20 0.40
RAB9A P51151 2/20 0.40
POLB P06746 2/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237756 0.87 HDAC3 (0.50) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL1064516 0.87 HDAC4 (0.62) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL3235060 0.82 KDM4E (0.38) HDAC3HDAC1GAAALDH1A1NPC1
SCHEMBL3262232 0.80 HDAC1 (0.39) HDAC3HDAC1HDAC2PKM
SCHEMBL3228530 0.80 HDAC1 (0.74) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL3234097 0.78 HDAC1 (0.48) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL3237174 0.78 HDAC1 (0.41) HDAC3HDAC1HDAC4HDAC2MEF2D
SCHEMBL3238636 0.76 HDAC3 (0.36) HDAC3HDAC1HDAC8HDAC6
SCHEMBL3241863 0.76 HDAC1 (0.52) HDAC3HDAC1HDAC4HDAC7HDAC2
SCHEMBL3238553 0.73 HDAC1 (0.44) HDAC3HDAC1HDAC2HDAC10HDAC11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028193-A1 COMPOUNDS INCLUDING PIMELIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO claimed